Cardiotonic effects of anthopleurin-A (AP-A), a polypeptide from a sea anemone, in dogs with a coronary artery stenosis. Eur J Pharmacol 1985 Apr 02;110(2):271-6
Date
04/02/1985Pubmed ID
3987818DOI
10.1016/0014-2999(85)90223-7Scopus ID
2-s2.0-0021814522 (requires institutional sign-in at Scopus site) 19 CitationsAbstract
The positive inotropic effect of AP-A was studied in anesthetized dogs with a severe stenosis of the left anterior descending coronary artery. Peak positive dP/dt (mm Hg/s) and % segment shortening (%SS) were used as indices of contractile function. AP-A (1.5-5.0 micrograms/kg, i.v.) produced positive inotropic effects globally (dP/dt, 1700 +/- 100 to 2650 +/- 250 mm Hg/s) and locally in the ischemic zone (%SS, 6.7 +/- 1.7 to 13.7 +/- 1.5%) without changing heart rate, mean arterial pressure or myocardial blood flow. These data suggest that AP-A may be potentially useful in the management of heart failure.
Author List
Gross GJ, Warltier DC, Hardman HF, Shibata SAuthor
David C. Warltier PhD Emeritus Professor in the Anesthesiology department at Medical College of WisconsinMESH terms used to index this publication - Major topics in bold
AnimalsBlood Pressure
Cardiotonic Agents
Coronary Circulation
Coronary Disease
Dogs
Female
Heart Rate
Intercellular Signaling Peptides and Proteins
Male
Myocardial Contraction
Peptides









